SCHEMBL9527288

SCHEMBL9527288

Cc1cccnc1C[S+]([O-])c1nc2cc(OC(F)(F)F)c(C(F)(F)F)cc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 4/20 0.33
S1PR2 O95136 2/20 0.33
RUNX1 Q01196 4/20 0.32
CBFB Q13951 2/20 0.32
CACNA1H O95180 1/20 0.32
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527817 0.89 ATP4A (0.36) RUNX1CBFB
SCHEMBL9529518 0.87 ATP4A (0.35) S1PR2RUNX1CBFB
SCHEMBL9531496 0.85 ATP4A (0.42) S1PR2RUNX1CACNA1H
SCHEMBL9527334 0.83 CBFB (0.40) TRPV1RUNX1CBFB
SCHEMBL9531500 0.81 ATP4A (0.44) CBFB
SCHEMBL10713063 0.80 KIF11 (0.39) TRPV1CBFB
SCHEMBL10713068 0.80 DYRK1A (0.46) TRPV1CBFB
SCHEMBL9526251 0.79 ATP4A (0.38) TRPV1
SCHEMBL9526628 0.79 CYP1A2 (0.48)
SCHEMBL9527662 0.78 RUNX1 (0.33) RUNX1CBFB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0134400-B1 FLUOROALKOXYSUBSTITUTED PYRIDYLMETHYLTHIO-(OR SULFINYL-)BENZIMIDAZOLES HAVING A SECRETOLYTIC ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1993-03-24 EP disclosed
US-4555518-A ANTIULCER AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1985-11-26 US disclosed
EP-0134400-A2 Fluoroalkoxysubstituted pyridylmethylthio-(or sulfinyl-)benzimidazoles having a secretolytic activity Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1985-03-20 EP disclosed