SCHEMBL9527504

SCHEMBL9527504

O=c1c([N+](=O)[O-])c[nH]n1-c1c(Cl)cc(C(F)(F)F)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
TDP1 Q9NUW8 3/20 0.50
ALDH1A1 P00352 2/20 0.50
TSHR P16473 2/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
HIF1A Q16665 1/20 0.50
TXNRD1 Q16881 1/20 0.50
TXNRD3 Q86VQ6 1/20 0.50
TXNRD2 Q9NNW7 1/20 0.50
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.40
PLK1 P53350 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PTPN5 P54829 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10444731 0.75 CYP3A4 (0.55) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL7819749 0.71 ALDH1A1 (0.82) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL10444468 0.70 CYP3A4 (0.45) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL9730621 0.70 CYP3A4 (0.47) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL10444826 0.70 ALDH1A1 (0.48) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL10654236 0.69 CYP3A4 (0.50) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL9526043 0.69 TDP1 (0.50) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL29805021 0.69 CYP3A4 (0.68) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL1531127 0.69 CYP3A4 (0.68) CYP3A4TDP1ALDH1A1TSHRHPGD
SCHEMBL9530253 0.69 GABRB3 (0.40) CDK4CCND1GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0257296-B1 4-CYANO(NITRO)-5-OXY(THIO)-PYRAZOLE DERIVATIVES BAYER AG (DE) 1993-05-12 EP disclosed
US-4770692-A 4-cyano(nitro)-5-oxy(thio)-pyrazole derivatives, composition containing them, and herbicidal and plant growth regulating methods of using them BAYER AKTIENGESELLSCHAFT (DE) 1988-09-13 US disclosed
EP-0257296-A1 4-Cyano(nitro)-5-oxy(thio)-pyrazole derivatives BAYER AG (DE) 1988-03-02 EP disclosed