SCHEMBL9530253

SCHEMBL9530253

O=c1cc[nH]n1-c1c(Cl)cc(C(F)(F)F)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRB3 P28472 9/20 0.40
GABRA2 P47869 7/20 0.38
GABRB2 P47870 7/20 0.38
GABRP O00591 3/20 0.38
GABRD O14764 3/20 0.38
GABRA1 P14867 3/20 0.38
GABRB1 P18505 3/20 0.38
GABRG2 P18507 3/20 0.38
GABRA5 P31644 3/20 0.38
GABRA3 P34903 3/20 0.38
GABRA4 P48169 3/20 0.38
GABRE P78334 3/20 0.38
GABRA6 Q16445 3/20 0.38
GABRG1 Q8N1C3 3/20 0.38
GABRG3 Q99928 3/20 0.38
GABRQ Q9UN88 3/20 0.38
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
MAPK14 Q16539 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10883634 0.81 MEN1 (0.37) CDK4CCND1HSD17B10
SCHEMBL9727098 0.76 GABRA2 (0.40) GABRB3GABRA2GABRB2GABRPGABRD
SCHEMBL9727138 0.76 ALDH1A1 (0.49) GABRB3GABRA2GABRB2GABRPGABRD
SCHEMBL10565417 0.74 ALDH1A1 (0.48) GABRB3GABRA2GABRB2GABRPGABRD
SCHEMBL9194415 0.73 GABRB3 (0.39) GABRB3GABRA2GABRB2GABRPGABRD
SCHEMBL10946405 0.73 TRPV1 (0.53) RAD51
SCHEMBL9194934 0.70 GABRP (0.46) GABRB3GABRA2GABRB2GABRPGABRD
SCHEMBL10679158 0.69 GABRA2 (0.38) GABRB3GABRA2GABRB2GABRPGABRD
SCHEMBL9527504 0.69 CYP3A4 (0.50) GABRB3CDK4CCND1
SCHEMBL9727104 0.69 P2RX1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1042937-C Substituted fused pyrazolo compounds and their use as herbicides ZENECA LTD (GB) 1999-04-14 CN disclosed
EP-0257296-B1 4-CYANO(NITRO)-5-OXY(THIO)-PYRAZOLE DERIVATIVES BAYER AG (DE) 1993-05-12 EP disclosed
US-5162528-A Pre- and post-emergence; phytaphthora in tomato plants; rice and wheat BAYER AKTIENGESELLSCHAFT (DE) 1992-11-10 US disclosed
US-5028717-A Herbicidal and fungicidal agents based on substituted pyrazolin-5-one derivatives BAYER AKTIENGESELLSCHAFT (DE) 1991-07-02 US disclosed
US-4909827-A Containing a C6-10 aryl group substituted in position 1 BAYER AKTIENGESELLSCHAFT (DE) 1990-03-20 US disclosed
US-4804398-A 1-aryl-4-cyano-5-halogenopyrazoles, composition containing them, and method of using them as selective herbicides BAYER AKTIENGESELLSCHAFT (DE) 1989-02-14 US disclosed
US-4770692-A 4-cyano(nitro)-5-oxy(thio)-pyrazole derivatives, composition containing them, and herbicidal and plant growth regulating methods of using them BAYER AKTIENGESELLSCHAFT (DE) 1988-09-13 US disclosed
EP-0257296-A1 4-Cyano(nitro)-5-oxy(thio)-pyrazole derivatives BAYER AG (DE) 1988-03-02 EP disclosed