SCHEMBL9528653

SCHEMBL9528653

CCCCCN1CCCC(COc2ccc(Cc3ccccc3)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.53
LTA4H P09960 9/20 0.51
CHRNB2 P17787 3/20 0.48
CHRNB4 P30926 3/20 0.48
CHRNA3 P32297 3/20 0.48
CHRNA4 P43681 3/20 0.48
CARM1 Q86X55 1/20 0.47
PRMT6 Q96LA8 1/20 0.47
KCNH2 Q12809 1/20 0.47
MAOA P21397 2/20 0.46
ACHE P22303 2/20 0.46
MAOB P27338 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9529213 0.99 HRH3 (0.52) HRH3LTA4HCHRNB2CHRNB4CHRNA3
SCHEMBL9368468 0.93 LTA4H (0.58) HRH3LTA4HCARM1PRMT6KCNH2
Hydrochloric Acid SCHEMBL27342609 0.92 CHRNB4 (0.50) HRH3LTA4HCHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL9372841 0.92 LTA4H (0.57) HRH3LTA4HCARM1PRMT6KCNH2
SCHEMBL9527422 0.91 KDM4E (0.54) HRH3LTA4HCHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL9527542 0.90 KDM4E (0.53) HRH3LTA4HCHRNB2CHRNB4CHRNA3
SCHEMBL9531944 0.89 HRH3 (0.61) HRH3CHRNB2CHRNB4CHRNA3CHRNA4
Oxalic Acid SCHEMBL9528802 0.86 KDM4E (0.54) HRH3CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9368505 0.86 KCNH2 (0.55) HRH3LTA4HKCNH2
Oxalic Acid SCHEMBL9697600 0.85 CHRNB2 (0.58) HRH3CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542844-A1 3-SUBSTITUTED PIPERIDINE DERIVATIVES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-05-26 EP claimed
WO-1992002501-A1 3-SUBSTITUTED PIPERIDINE DERIVATIVES SMITHKLINE & FRENCH LABORATORIES LIMITED (GB) 1992-02-20 WO claimed
WO-1992002501-A1 3-SUBSTITUTED PIPERIDINE DERIVATIVES SMITHKLINE & FRENCH LABORATORIES LIMITED (GB) 1992-02-20 WO disclosed