SCHEMBL9529209

SCHEMBL9529209

Cc1nc2c(OCCc3ccccc3)cccc2[nH]1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.71
DRD4 P21917 3/20 0.71
DRD3 P35462 3/20 0.71
CBFB Q13951 2/20 0.43
IDO1 P14902 1/20 0.42
DHODH Q02127 3/20 0.41
CYP11B1 P15538 3/20 0.41
CYP11B2 P19099 3/20 0.41
PARP1 P09874 1/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
MAOA P21397 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7619109 0.86 DRD2 (0.67) DRD2DRD4DRD3CBFBDHODH
SCHEMBL8126835 0.83 DRD4 (1.00) DRD2DRD4DRD3
SCHEMBL13165012 0.80 DRD2 (0.60) DRD2DRD4DRD3CBFBPARP1
SCHEMBL6510308 0.78 DRD2 (0.49) DRD2DRD4DRD3CBFBPARP1
SCHEMBL9529218 0.78 DRD2 (0.45) DRD2DRD4DRD3IDO1CYP11B1
SCHEMBL9528482 0.78 MEN1 (0.59) DRD2DRD4DRD3CBFBDHODH
SCHEMBL7612954 0.74 DRD2 (0.53) DRD2DRD4DRD3CBFBDHODH
SCHEMBL9528411 0.74 DRD2 (0.53) DRD2DRD4DRD3CBFBDHODH
SCHEMBL6510296 0.74 DRD2 (0.45) DRD2DRD4DRD3CBFBPARP1
SCHEMBL4611125 0.74 ALDH1A1 (0.55) DRD2DRD4DRD3CBFBDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266326-B1 NOVEL DERIVATIVES OF BENZIMIDAZOLES ACTIVE AS ANTI-ULCER AGENTS Aktiebolaget Hässle (SE) 1993-03-10 EP disclosed
US-5106862-A DERIVATIVES OF BENZIMIDAZOLES ACTIVE AS ANTI-ULCER AGENTS AKTIEBOLAGET HASSLE (SE) 1992-04-21 US disclosed
EP-0266326-A1 Novel derivatives of benzimidazoles active as anti-ulcer agents Aktiebolaget Hässle (SE) 1988-05-04 EP disclosed