SCHEMBL9529217

SCHEMBL9529217

CCCNCC1CN(c2ccccc2)c2ccccc2O1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.61
POLB P06746 1/20 0.58
ESR2 Q92731 1/20 0.58
CASR P41180 4/20 0.55
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
GRM2 Q14416 5/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9455126 0.99 HTR1A (0.60) HTR1APOLBESR2CASRADRA1D
SCHEMBL9532833 0.83 CASR (0.59) HTR1ACASRADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL9455227 0.82 CASR (0.58) HTR1ACASRADRA1DADRA1AADRA1B
SCHEMBL9455114 0.76 CASR (0.50) HTR1ACASRADRA1DADRA1AADRA1B
SCHEMBL6977935 0.76 CASR (0.50) HTR1ACASRADRA1DADRA1AADRA1B
SCHEMBL9529252 0.76 CASR (0.50) HTR1ACASRADRA1DADRA1AADRA1B
Fumaric Acid SCHEMBL9455274 0.75 MAPT (0.45) HTR1APOLBESR2CASR
SCHEMBL6969866 0.75 HTR1A (1.00) HTR1ACASR
SCHEMBL10864903 0.75 POLB (0.97) HTR1APOLBESR2ADRA1DADRA1A
SCHEMBL29353196 0.75 POLB (0.97) HTR1APOLBESR2ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359790-B1 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5084454-A Tranquilizers and antinausea drugs FARMITALIA CARLO ERBA S.R.L. (IT) 1992-01-28 US disclosed