SCHEMBL9532833

SCHEMBL9532833

CNCC1CN(c2ccccc2)c2ccccc2O1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASR P41180 10/20 0.59
HTR1A P08908 3/20 0.54
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
GRM2 Q14416 3/20 0.42
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9455227 0.99 CASR (0.58) CASRHTR1AADRA1DADRA1AADRA1B
SCHEMBL9529217 0.83 HTR1A (0.61) CASRHTR1AADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL9455126 0.82 HTR1A (0.60) CASRHTR1AADRA1DADRA1AADRA1B
SCHEMBL6977935 0.80 CASR (0.50) CASRHTR1AADRA1DADRA1AADRA1B
SCHEMBL9529252 0.80 CASR (0.50) CASRHTR1AADRA1DADRA1AADRA1B
SCHEMBL9455114 0.80 CASR (0.50) CASRHTR1AADRA1DADRA1AADRA1B
SCHEMBL9699321 0.79 HTR6 (0.43) CASRHTR1AADRA1AHTR6
Hydrochloric Acid SCHEMBL9455268 0.79 CASR (0.49) CASRHTR1AGRM2
SCHEMBL9701358 0.75 HTR6 (0.41) CASRHTR1AADRA1AHTR6
SCHEMBL12614493 0.75 CASR (1.00) CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359790-B1 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5084454-A Tranquilizers and antinausea drugs FARMITALIA CARLO ERBA S.R.L. (IT) 1992-01-28 US disclosed
EP-0359790-A1 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION. ERBA CARLO SPA (IT) 1990-03-28 EP disclosed
WO-1989007596-A1 NEW 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-08-24 WO disclosed