SCHEMBL9530568

SCHEMBL9530568

CC1(C)C=C(C(=O)Cl)c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 4/20 0.34
APEX1 P27695 1/20 0.33
KMT2A Q03164 2/20 0.33
ITGA4 P13612 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
S100A4 P26447 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
PDK2 Q15119 2/20 0.32
NOTUM Q6P988 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31563811 0.70 PDK2 (0.35) THRBTDP1ALDH1A1KMT2AMEN1
SCHEMBL22172193 0.70 PDK2 (0.34) TDP1ALDH1A1ITGA4S100A4PDK2
SCHEMBL7258801 0.69 APOBEC3A (0.48) TDP1ALDH1A1KMT2AITGA4MEN1
SCHEMBL29374343 0.69 APOBEC3A (0.48) TDP1ALDH1A1KMT2AITGA4MEN1
SCHEMBL30888607 0.68 THRB (0.47) THRBTDP1ALDH1A1APEX1KMT2A
SCHEMBL9938667 0.68 THRB (0.47) THRBTDP1ALDH1A1APEX1KMT2A
SCHEMBL23292666 0.66 KDM4E (0.38) TDP1ALDH1A1KMT2AITGA4MEN1
SCHEMBL29840752 0.66 KDM4E (0.38) TDP1ALDH1A1KMT2AITGA4MEN1
SCHEMBL11294332 0.66 S100A4 (0.33) THRBTDP1ALDH1A1KMT2AITGA4
SCHEMBL4636505 0.66 THRB (0.48) THRBTDP1ALDH1A1APEX1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289170-B1 AZABICYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1993-06-23 EP disclosed
US-4882327-A NERVOUS SYSTEM DISORDERS BEECHAM GROUP P.L.C. (GB) 1989-11-21 US disclosed
EP-0289170-A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-11-02 EP disclosed