SCHEMBL9533336

SCHEMBL9533336

Cc1csc2nc3c(Cl)cccc3c(=O)n12

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.62
HSD17B10 Q99714 4/20 0.62
ALDH1A1 P00352 4/20 0.62
HPGD P15428 3/20 0.62
SMN1; SMN2 Q16637 1/20 0.51
RCE1 Q9Y256 1/20 0.51
GLA P06280 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
TSHR P16473 1/20 0.46
PARP1 P09874 1/20 0.44
MAPT P10636 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PDE7A Q13946 1/20 0.41
PIK3CD O00329 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9532194 0.86 KDM4E (0.65) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL10696506 0.83 ALDH1A1 (0.62) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL9536686 0.81 KDM4E (0.59) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL9536068 0.80 KDM4E (0.50) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL9533007 0.78 ALDH1A1 (0.55) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL9533630 0.78 KDM4E (0.62) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL10696216 0.78 PARP1 (0.44) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL10978164 0.77 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL10696717 0.76 PARP1 (0.43) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2
SCHEMBL9533620 0.75 KDM4E (0.48) KDM4EHSD17B10ALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0263523-B1 Process for the preparation of thiazolo [2,3-b] quinazolones BASF AG (DE) 1993-12-29 EP claimed
EP-0263523-A2 Process for the preparation of thiazolo [2,3-b] quinazolones BASF Aktiengesellschaft (DE) 1988-04-13 EP claimed
EP-0263523-B1 Process for the preparation of thiazolo [2,3-b] quinazolones BASF AG (DE) 1993-12-29 EP disclosed
US-5030727-A Reacting an anthronilide derivative with a thiazole derivative or a fluorozuinazolone with a neucleophile BASF AKTIENGESELLSCHAFT (DE) 1991-07-09 US disclosed
EP-0263523-A2 Process for the preparation of thiazolo [2,3-b] quinazolones BASF Aktiengesellschaft (DE) 1988-04-13 EP disclosed
EP-0263523-A2 Process for the preparation of thiazolo [2,3-b] quinazolones BASF Aktiengesellschaft (DE) 1988-04-13 EP disclosed