SCHEMBL9533499

SCHEMBL9533499

CN1C2CCC1CC(NC(=O)C1=CC(C)(C)c3ccccc31)C2

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 1/20 0.48
CYP3A4 P08684 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
HSD17B10 Q99714 1/20 0.48
HTR3A P46098 5/20 0.46
HTR3E A5X5Y0 3/20 0.46
HTR3B O95264 3/20 0.46
HTR3D Q70Z44 3/20 0.46
HTR3C Q8WXA8 3/20 0.46
SLC22A2 O15244 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44
KCNH2 Q12809 1/20 0.44
SLC47A1 Q96FL8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9531070 0.86 HPGD (0.37) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL1559634 0.74 MEN1 (0.74) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL9531125 0.73 CHRM2 (0.59) HTR3AHTR3EHTR3BHTR3DHTR3C
Hydrochloric Acid SCHEMBL9533193 0.72 CHRM2 (0.58) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9532593 0.72 GAA (0.59) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL9533289 0.71 HTR3A (0.55) MEN1KMT2AALDH1A1CYP3A4TSHR
Hydrochloric Acid SCHEMBL9533542 0.70 HTR3A (0.54) MEN1KMT2AALDH1A1CYP3A4TSHR
SCHEMBL3533984 0.69 GAA (0.68) MEN1KMT2AALDH1A1CYP3A4TSHR
Ricasetron SCHEMBL21715163 0.69 NOTUM (0.52) HTR3A
Ricasetron SCHEMBL634827 0.69 NOTUM (0.52) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289170-B1 AZABICYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1993-06-23 EP claimed
EP-0289170-A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-11-02 EP claimed