SCHEMBL9534700

SCHEMBL9534700

CSC(=NC(C)C(C)(C)C)NC#N

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 5/20 0.49
KCNJ11 Q14654 5/20 0.49
ALDH1A1 P00352 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
ALOX15 P16050 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPK1 P28482 1/20 0.47
HIF1A Q16665 1/20 0.47
HSD17B10 Q99714 1/20 0.47
LMNA P02545 1/20 0.47
GLA P06280 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.36
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11542408 0.74 ALDH1A1 (0.42) ABCC9KCNJ11ALDH1A1CYP1A2CYP2C9
SCHEMBL11542404 0.74 ALDH1A1 (0.42) ABCC9KCNJ11ALDH1A1CYP1A2CYP2C9
SCHEMBL9534597 0.72 ALDH1A1 (0.47) ABCC9KCNJ11ALDH1A1CYP1A2CYP2C9
SCHEMBL4477801 0.69
SCHEMBL4477799 0.69
SCHEMBL11162280 0.67 ABCC9 (0.47) ABCC9KCNJ11ALDH1A1CYP3A4CYP1A2
SCHEMBL11509173 0.67 ALDH1A1 (0.42) ABCC9KCNJ11ALDH1A1SMN1; SMN2
SCHEMBL11087993 0.64
SCHEMBL11087989 0.64
Pinacidil Anhydrous SCHEMBL1650693 0.64 ABCC9 (1.00) ABCC9KCNJ11ALDH1A1CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377528-B1 Piperidines, process for their preparation and pharmaceutical compounds containing them LIPHA (FR) 1993-12-08 EP disclosed
US-5001134-A Piperidines, processes of preparation and medications containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1991-03-19 US disclosed
EP-0377528-A1 Piperidines, process for their preparation and pharmaceutical compounds containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1990-07-11 EP disclosed