SCHEMBL9534725

SCHEMBL9534725

COc1cc(-c2ccc3ccccc3c2)ccc1C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.66
ALDH1A1 P00352 4/20 0.66
HPGD P15428 3/20 0.66
ACMSD Q8TDX5 1/20 0.58
CHEK1 O14757 1/20 0.55
ERN1 O75460 1/20 0.55
APAF1 O14727 1/20 0.54
RECQL P46063 1/20 0.54
CASP6 P55212 1/20 0.54
CACNA1B Q00975 1/20 0.54
APBA1 Q02410 1/20 0.54
MCL1 Q07820 1/20 0.54
CASP8 Q14790 1/20 0.54
HSD17B10 Q99714 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23143203 0.88 KDM4E (0.66) KDM4EALDH1A1HPGDACMSDERN1
SCHEMBL504872 0.87 CHEK1 (0.60) KDM4EALDH1A1HPGDACMSDCHEK1
SCHEMBL29788086 0.87 CHEK1 (0.60) KDM4EALDH1A1HPGDACMSDCHEK1
SCHEMBL2770512 0.87 ALDH1A1 (0.67) KDM4EALDH1A1HPGDCHEK1APAF1
SCHEMBL14156931 0.86 ESR1 (0.56) KDM4EALDH1A1HPGDACMSDCHEK1
SCHEMBL8692896 0.84 KDM4E (0.49) KDM4EALDH1A1HPGDCHEK1APAF1
SCHEMBL17177740 0.83 ALDH1A1 (0.62) KDM4EALDH1A1HPGDCHEK1APAF1
SCHEMBL10459347 0.82 ALDH1A1 (0.61) KDM4EALDH1A1HPGDCHEK1APAF1
SCHEMBL617928 0.80 ALDH1A1 (1.00) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL9537888 0.80 MCL1 (0.62) KDM4EALDH1A1HPGDACMSDCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532531-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-03-24 EP disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed