SCHEMBL9534890

SCHEMBL9534890

Cn1cc2c(n1)-c1cnn(C)c1CS2

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.40
PLK1 P53350 1/20 0.35
CSNK2A1 P68400 1/20 0.35
PLK3 Q9H4B4 1/20 0.35
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538656 0.73 PLK1 (0.39) PLK1CSNK2A1PLK3
SCHEMBL9220489 0.71 DRD4 (0.47) MMP12PLK1CSNK2A1PLK3
SCHEMBL9534036 0.69 CSNK2A1 (0.35) PLK1CSNK2A1PLK3
SCHEMBL9216050 0.69 DRD4 (0.56) MMP12PLK1CSNK2A1PLK3
SCHEMBL9214111 0.68 PLK1 (0.34) PLK1CSNK2A1PLK3
SCHEMBL9534430 0.61 PLK1 (0.56) PLK1CSNK2A1PLK3
SCHEMBL9535703 0.61 PLK1 (0.61) PLK1CSNK2A1PLK3
SCHEMBL9534532 0.60 PLK1 (0.54) PLK1CSNK2A1PLK3
Hydrochloric Acid SCHEMBL9534437 0.59 PLK1 (0.59) PLK1CSNK2A1PLK3
SCHEMBL9533936 0.58 PLK1 (0.74) PLK1CSNK2A1PLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276835-B1 PYRAZOLOTHIOPYRANOPYRAZOLES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-03-17 EP disclosed
EP-0276835-A1 Pyrazolothiopyranopyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734431-A Thiopyranodipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed