SCHEMBL9538656

SCHEMBL9538656

Cn1ncc2c1CSc1cnn(C)c1-2

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.39
CSNK2A1 P68400 1/20 0.39
PLK3 Q9H4B4 1/20 0.39
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9534036 0.73 CSNK2A1 (0.35) PLK1CSNK2A1PLK3
SCHEMBL9211095 0.67 PLK1 (0.49) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL9534430 0.66 PLK1 (0.56) PLK1CSNK2A1PLK3DRD2HIF1A
Hydrochloric Acid SCHEMBL9216167 0.66 PLK1 (0.47) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL9535703 0.65 PLK1 (0.61) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL10798104 0.65 DRD2 (0.47) DRD2DRD4HIF1A
Hydrochloric Acid SCHEMBL9534437 0.63 PLK1 (0.59) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL19153460 0.63 PLK1 (0.44) PLK1CSNK2A1PLK3DRD2DRD4
SCHEMBL10368994 0.61 MMP12 (0.57) DRD2DRD4
SCHEMBL9211138 0.59 PLK1 (0.44) PLK1CSNK2A1PLK3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276835-B1 PYRAZOLOTHIOPYRANOPYRAZOLES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-03-17 EP disclosed
US-4734431-A Thiopyranodipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed