SCHEMBL9535409

SCHEMBL9535409

O=c1ccc2c(OCC3CO3)cccc2o1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.62
CYP3A4 P08684 4/20 0.58
KCNA3 P22001 3/20 0.56
ALDH1A1 P00352 4/20 0.49
GLA P06280 2/20 0.49
ALOX15 P16050 2/20 0.47
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44
TDP1 Q9NUW8 1/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39
KCNA5 P22460 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
MAOB P27338 1/20 0.36
NCOA1 Q15788 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8623175 0.78 MAOA (0.57) CYP3A4ALDH1A1GLATP53TSHR
SCHEMBL729501 0.78 ALDH1A1 (0.65) CYP3A4ALDH1A1GLATP53TSHR
SCHEMBL6309685 0.78 ALDH1A1 (0.53) CYP2A6CYP3A4KCNA3ALDH1A1GLA
SCHEMBL6309690 0.78 ALDH1A1 (0.53) CYP2A6CYP3A4KCNA3ALDH1A1GLA
SCHEMBL7966131 0.78 ALDH1A1 (0.53) CYP2A6CYP3A4KCNA3ALDH1A1GLA
SCHEMBL11036109 0.77 CYP2A6 (1.00) CYP2A6CYP3A4KCNA3ALDH1A1GLA
SCHEMBL5432111 0.77 ALDH1A1 (0.56) CYP2A6CYP3A4ALDH1A1GLATP53
SCHEMBL6317536 0.77 ALDH1A1 (0.56) CYP2A6CYP3A4ALDH1A1GLATP53
SCHEMBL13007252 0.77 MCL1 (0.53) CYP3A4ALDH1A1GLAALOX15TP53
SCHEMBL13061433 0.77 MCL1 (0.53) CYP3A4ALDH1A1GLAALOX15TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5254595-A Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them ELF SANOFI (FR) 1993-10-19 US disclosed
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed