SCHEMBL9535904

SCHEMBL9535904

Fc1ccc(Cn2c(CC3CCNCC3)nc3ccncc32)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.54
ENPP2 Q13822 1/20 0.48
NR4A2 P43354 1/20 0.47
HPGD P15428 2/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.44
NLRP3 Q96P20 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
HTR3A P46098 1/20 0.43
RAB9A P51151 1/20 0.43
CHRM1 P11229 1/20 0.43
HRH1 P35367 1/20 0.43
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL10553663 0.92 ENPP2 (0.48) KCNH2ENPP2NR4A2HPGDTP53
SCHEMBL9538624 0.85 KCNH2 (0.63) KCNH2NR4A2HTR3ARAB9ACHRM1
SCHEMBL9382803 0.85 KCNH2 (0.64) KCNH2NR4A2HTR3ARAB9ACHRM1
SCHEMBL9538842 0.83 SSTR5 (0.52) ENPP2RAB9A
SCHEMBL9537733 0.83 ENPP2 (0.44) ENPP2HPGDTP53MAPTLMNA
SCHEMBL9535886 0.82 KCNH2 (0.59) KCNH2NR4A2HTR3ARAB9ACHRM1
SCHEMBL9565088 0.82 KCNH2 (0.48) KCNH2NR4A2HPGDLMNAHTR3A
SCHEMBL9564851 0.80 CYP1A2 (0.54) KCNH2NR4A2HPGDLMNASMN1; SMN2
SCHEMBL9537437 0.80 KCNH2 (0.59) KCNH2NR4A2HTR3ACHRM1HRH1
SCHEMBL9540203 0.80 KCNH2 (0.64) KCNH2NR4A2HTR3ARAB9ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed