SCHEMBL9536060

SCHEMBL9536060

Fc1ccc(N2CCN(CCCCl)CC2)c(F)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 4/20 0.60
HTR1A P08908 5/20 0.52
ADRA1A P35348 4/20 0.52
ADRA1D P25100 3/20 0.52
HTR7 P34969 3/20 0.51
HTR6 P50406 2/20 0.51
SLC6A2 P23975 1/20 0.51
SLC6A3 Q01959 1/20 0.51
KCNH2 Q12809 2/20 0.49
PARP1 P09874 1/20 0.49
PARP2 Q9UGN5 1/20 0.49
PTGS2 P35354 1/20 0.47
LMNA P02545 2/20 0.44
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 1/20 0.44
NLRP1 Q9C000 1/20 0.44
DRD3 P35462 2/20 0.43
DRD2 P14416 1/20 0.43
DRD1 P21728 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10573066 0.98 ADRA1B (0.62) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL5836414 0.91 ADRA1B (0.55) ADRA1BHTR1AADRA1AADRA1DHTR7
Hydrochloric Acid SCHEMBL10574990 0.89 ADRA1B (0.57) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL4910280 0.85 ADRA1B (0.63) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL9536914 0.85 ADRA1B (0.60) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL8146772 0.85 PTGS2 (0.62) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL8151383 0.84 ADRA1B (0.62) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL22125822 0.83 ADRA1B (0.56) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL13321530 0.82 ADRA1B (0.60) ADRA1BHTR1AADRA1AADRA1DHTR7
SCHEMBL28739481 0.82 LMNA (0.60) ADRA1BHTR1AADRA1AADRA1DHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254623-B1 AMINOALKYLTHIO TRIAZOLOPYRIDINE OR TRIAZOLOQUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM, PARTICULARLY USEFUL AS ANTALGICS LABORATOIRES UPSA (FR) 1993-06-09 EP disclosed
US-4886805-A Novel aminoalkylthio derivatives of triazolopyridine or triazoloquinoline, the processes for their preparation, and drugs, useful especially as analgesics, in which they are present Centre D'Activite Et De Recherches Pharmaceutique Industrielle Biologique Medicale (FR) 1989-12-12 US disclosed
EP-0254623-A1 Aminoalkylthio triazolopyridine or triazoloquinoline derivatives, process for their preparation, medicaments containing them, particularly useful as antalgics LABORATOIRES UPSA (FR) 1988-01-27 EP disclosed