SCHEMBL9536078

SCHEMBL9536078

Fc1ccc(Cn2c(CC3CCNCC3)nc3ncccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.50
NR4A2 P43354 1/20 0.48
HTR3A P46098 1/20 0.44
HRH1 P35367 5/20 0.43
CHRM1 P11229 3/20 0.43
RAB9A P51151 1/20 0.41
CYP2D6 P10635 3/20 0.41
CYP3A4 P08684 2/20 0.41
PDE6D O43924 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL10554578 0.91 KCNH2 (0.43) KCNH2NR4A2HTR3AHRH1CHRM1
SCHEMBL9565088 0.85 KCNH2 (0.48) KCNH2NR4A2HTR3AHRH1CHRM1
SCHEMBL9382803 0.84 KCNH2 (0.64) KCNH2NR4A2HTR3AHRH1CHRM1
SCHEMBL9536547 0.84 SSTR5 (0.52) HTR3A
SCHEMBL9535735 0.83 TP53 (0.51) KCNH2NR4A2
SCHEMBL10804293 0.83 KCNH2 (0.47) KCNH2HRH1CHRM1RAB9ACYP2D6
Hydrochloric Acid SCHEMBL9537452 0.83 TP53 (0.50) KCNH2NR4A2
SCHEMBL9537190 0.82 PRMT3 (0.44) KCNH2HRH1CHRM1CYP2D6
SCHEMBL9538624 0.80 KCNH2 (0.63) KCNH2NR4A2HTR3AHRH1CHRM1
SCHEMBL9535904 0.79 KCNH2 (0.54) KCNH2NR4A2HTR3AHRH1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed