SCHEMBL9536348

SCHEMBL9536348

c1cc2c(c(OCC3CO3)c1)CCC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
GLA P06280 1/20 0.54
TP53 P04637 1/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HIF1A Q16665 1/20 0.49
RXRB P28702 9/20 0.48
RXRA P19793 9/20 0.48
RXRG P48443 6/20 0.48
TDP1 Q9NUW8 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.46
SSTR4 P31391 1/20 0.41
HTR2A P28223 3/20 0.40
SLC6A4 P31645 3/20 0.40
SLC6A2 P23975 1/20 0.39
HRH1 P35367 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7770798 0.97 ALDH1A1 (0.54) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL30974571 0.97 ALDH1A1 (0.54) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL9311184 0.92 ALDH1A1 (0.56) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL7769212 0.84 RXRA (0.44) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL11090866 0.81 ALDH1A1 (0.48) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL21254625 0.81 HTR2A (0.66) CYP3A4RXRBRXRARXRGHTR2A
SCHEMBL8432284 0.81 HTR2A (0.66) CYP3A4RXRBRXRARXRGHTR2A
SCHEMBL11514478 0.80 ALDH1A1 (0.47) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL9323483 0.79 ALDH1A1 (0.53) ALDH1A1GLATP53CYP3A4TSHR
SCHEMBL8051434 0.79 MRGPRX4 (0.52) ALDH1A1GLATP53CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5254595-A Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them ELF SANOFI (FR) 1993-10-19 US disclosed
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed