SCHEMBL9537104

SCHEMBL9537104

COC(=O)CC(N)C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.44
ALDH1A1 P00352 1/20 0.41
KIF11 P52732 10/20 0.41
KCNA5 P22460 1/20 0.40
POLB P06746 1/20 0.40
SLC7A5 Q01650 1/20 0.39
KMT2A Q03164 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27508043 0.79 KMT2A (0.45) KCNN4ALDH1A1KIF11KCNA5POLB
SCHEMBL1277655 0.74 KIF11 (0.58) KIF11
SCHEMBL1144412 0.74 ALDH1A1 (0.51) ALDH1A1KCNA5POLBKMT2ACYP1A2
SCHEMBL167043 0.74 ALDH1A1 (0.51) ALDH1A1KCNA5POLBKMT2ACYP1A2
SCHEMBL476790 0.74 ALDH1A1 (0.51) ALDH1A1KCNA5POLBKMT2ACYP1A2
Hydrochloric Acid SCHEMBL1277652 0.73 KIF11 (0.56) KIF11
Hydrochloric Acid SCHEMBL1277658 0.73 KIF11 (0.56) KIF11
Hydrochloric Acid SCHEMBL2203097 0.72 ALDH1A1 (0.50) ALDH1A1KCNA5POLBKMT2ACYP1A2
Hydrochloric Acid SCHEMBL476789 0.72 ALDH1A1 (0.50) ALDH1A1KCNA5POLBKMT2ACYP1A2
Hydrochloric Acid SCHEMBL6373800 0.72 ALDH1A1 (0.50) ALDH1A1KCNA5POLBKMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0535192-A1 NOVEL DNA GYRASE INHIBITORS, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL PREPARATIONS CONTAINING SAME. HOFFMANN LA ROCHE (CH) 1993-04-07 EP disclosed