SCHEMBL9537201

SCHEMBL9537201

O=c1cccc(-c2cccc3ccccc23)[nH]1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.61
ALPL P05186 1/20 0.61
GAA P10253 1/20 0.61
NOTUM Q6P988 1/20 0.52
TYMP P19971 1/20 0.46
GSK3B P49841 2/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
PTPN1 P18031 1/20 0.43
PDE10A Q9Y233 1/20 0.43
ADK P55263 1/20 0.42
POLB P06746 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754369 0.81 NOTUM (0.48) KDM4EALPLGAANOTUMCA12
SCHEMBL9534937 0.75 KDM4E (0.50) KDM4EALPLGAATYMPGSK3B
SCHEMBL30602735 0.74 NOTUM (0.53) KDM4EGAANOTUMPOLBCA12
SCHEMBL2116388 0.74 CA12 (0.53) KDM4EALPLGAATYMPPTPN1
SCHEMBL509972 0.74 KDM4E (0.57) KDM4EALPLGAATYMPGSK3B
SCHEMBL11736368 0.74 KDM4E (0.61) KDM4EALPLGAATYMPGSK3B
SCHEMBL8535240 0.73 NOTUM (0.68) KDM4ENOTUMCA12CA1CA9
SCHEMBL8570718 0.73 KDM4E (0.51) KDM4EALPLGAATYMPGSK3B
SCHEMBL2289477 0.72 KDM4E (0.50) KDM4EALPLGAATYMPGSK3B
SCHEMBL9754547 0.72 MCL1 (0.55) KDM4EALPLGAATYMPPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104418853-B Substituted naphthyridines-2-ketonic compound, preparation method, purposes and pharmaceutical composition 北大方正集团有限公司 2016-09-07 CN disclosed
EP-0532531-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-03-24 EP disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed