SCHEMBL8570718

SCHEMBL8570718

O=c1[nH]c(-c2cccc3ccccc23)co1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
ALPL P05186 1/20 0.51
GAA P10253 1/20 0.51
TYMP P19971 1/20 0.43
GSK3B P49841 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
PTPN1 P18031 1/20 0.40
PDE10A Q9Y233 1/20 0.40
MCL1 Q07820 1/20 0.40
PARP1 P09874 1/20 0.39
ENPP3 O14638 1/20 0.39
ENPP1 P22413 1/20 0.39
POLB P06746 1/20 0.39
PIM1 P11309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3749102 0.74 KDM4E (0.54) KDM4EMCL1PARP1
SCHEMBL9360263 0.74 NPC1 (0.47) KDM4E
SCHEMBL509972 0.74 KDM4E (0.57) KDM4EALPLGAATYMPGSK3B
SCHEMBL9537201 0.73 KDM4E (0.61) KDM4EALPLGAATYMPGSK3B
SCHEMBL16664827 0.72 MPO (0.53) KDM4EGAAGSK3BCDK5CDK5R1
SCHEMBL31059216 0.69 KDR (0.53) KDM4EGSK3BPOLB
SCHEMBL9534937 0.68 KDM4E (0.50) KDM4EALPLGAATYMPGSK3B
SCHEMBL25302086 0.67 ALDH1A1 (0.59) KDM4EALPLGAAPTPN1POLB
SCHEMBL29350007 0.67 ALDH1A1 (0.59) KDM4EALPLGAAPTPN1POLB
SCHEMBL27953 0.67 ALDH1A1 (0.59) KDM4EALPLGAAPTPN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0425209-B1 Naphthyloxazolidone derivatives TANABE SEIYAKU CO (JP) 1995-05-10 EP claimed
US-5332754-A Antidepressant TANABE SEIYAKU CO., LTD. (JP) 1994-07-26 US claimed
US-5182296-A Antidepressants TANABE SEIYAKY CO., LTD. (JP) 1993-01-26 US claimed
EP-0425209-A2 Naphthyloxazolidone derivatives TANABE SEIYAKU CO., LTD. (JP) 1991-05-02 EP claimed
JP-10226646-A None JP disclosed
JP-5155772-A None JP disclosed
JP-10218772-A None JP disclosed
JP-H10226646-A THERAPEUTIC AGENT OF PARKINSONISM TANABE SEIYAKU CO LTD 1998-08-25 JP disclosed
JP-H10218772-A PREVENTIVE AND THERAPEUTIC AGENT FOR HYPOBULIA AND LOWERING OF SPONTANEITY DUE TO CEREBROVASCULAR ACCIDENT OR DEPRESSION SYSTEM TANABE SEIYAKU CO LTD 1998-08-18 JP disclosed
EP-0425209-B1 Naphthyloxazolidone derivatives TANABE SEIYAKU CO (JP) 1995-05-10 EP disclosed
EP-0425209-B1 Naphthyloxazolidone derivatives TANABE SEIYAKU CO (JP) 1995-05-10 EP disclosed
US-5332754-A Antidepressant TANABE SEIYAKU CO., LTD. (JP) 1994-07-26 US disclosed
US-5332754-A Antidepressant TANABE SEIYAKU CO., LTD. (JP) 1994-07-26 US disclosed
US-5332754-A Antidepressant TANABE SEIYAKU CO., LTD. (JP) 1994-07-26 US disclosed
JP-H05155772-A ANTIDEPRESSANT TANABE SEIYAKU CO LTD 1993-06-22 JP disclosed
US-5182296-A Antidepressants TANABE SEIYAKY CO., LTD. (JP) 1993-01-26 US disclosed
US-5182296-A Antidepressants TANABE SEIYAKY CO., LTD. (JP) 1993-01-26 US disclosed
EP-0425209-A2 Naphthyloxazolidone derivatives TANABE SEIYAKU CO., LTD. (JP) 1991-05-02 EP disclosed
EP-0425209-A2 Naphthyloxazolidone derivatives TANABE SEIYAKU CO., LTD. (JP) 1991-05-02 EP disclosed
EP-0425209-A2 Naphthyloxazolidone derivatives TANABE SEIYAKU CO., LTD. (JP) 1991-05-02 EP disclosed