SCHEMBL9537241

SCHEMBL9537241

N#CNc1c(F)cccc1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.38
ADORA2B P29275 2/20 0.38
ADORA2A P29274 2/20 0.38
HTT P42858 2/20 0.37
ALDH1A1 P00352 4/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
RAB9A P51151 2/20 0.35
LMNA P02545 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
DHODH Q02127 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
NFKB2 Q00653 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10512435 0.80 KMT2A (0.35) HTTALDH1A1KMT2AMEN1HPGD
SCHEMBL9311569 0.79 CYP2A6 (0.40) ADORA1ADORA2AHTTALDH1A1RAB9A
SCHEMBL18634828 0.76 ADORA2B (0.41) ADORA1ADORA2BHTTALDH1A1KMT2A
SCHEMBL6353571 0.72 ADORA1 (0.45) ADORA1ADORA2BADORA2AHTTALDH1A1
SCHEMBL9536942 0.72 PTGS2 (0.44) HTTALDH1A1KMT2ARAB9ALMNA
SCHEMBL421370 0.72 ADORA1 (0.51) ADORA1ADORA2BADORA2AALDH1A1KMT2A
SCHEMBL3911337 0.71 HTT (0.51) HTTALDH1A1KMT2AMEN1RAB9A
Hydrochloric Acid SCHEMBL29097687 0.71 MAPK1 (0.48) ADORA1ADORA2AHTTALDH1A1KMT2A
SCHEMBL9310587 0.71 FABP3 (0.43) HTTALDH1A1KMT2AMEN1LMNA
Hydrochloric Acid SCHEMBL28562921 0.69 MAPK1 (0.47) ADORA1ADORA2AHTTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0536151-A1 ORTHOSUBSTITUTED BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM. BOOTS CO PLC (GB) 1993-04-14 EP disclosed