SCHEMBL9537294

SCHEMBL9537294

Cc1cc(-c2cccc(C(F)(F)F)c2)c2nc(C(F)(F)F)nn2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KCNH2 Q12809 1/20 0.41
ADORA2A P29274 2/20 0.40
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
ADORA1 P30542 1/20 0.39
CYP17A1 P05093 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535623 0.76 PTGS2 (0.46) KDM4EHPGDHSD17B10ALDH1A1CYP1A2
SCHEMBL9534839 0.69 HSD17B10 (0.49) KDM4EHPGDHSD17B10ALDH1A1
SCHEMBL9535483 0.67 IKBKB (0.52) KDM4EHPGDHSD17B10ALDH1A1CYP1A2
SCHEMBL19987117 0.67 PIM1 (0.58) KDM4EHSD17B10ALDH1A1ADORA2AJAK2
SCHEMBL9056918 0.66 PTPN5 (0.48) KDM4EHPGDCYP1A2CYP3A4SMN1; SMN2
SCHEMBL1722035 0.66 NFKBIA (0.43) KDM4EHPGDALDH1A1TDP1ADORA2A
SCHEMBL11389842 0.66 JAK2 (0.45) KDM4EHPGDHSD17B10ALDH1A1CYP1A2
SCHEMBL21254035 0.66 NPC1 (0.54) HPGDALDH1A1CYP1A2CYP3A4KCNH2
SCHEMBL2615262 0.65 CTSS (0.60) KDM4EHPGDHSD17B10ALDH1A1CYP1A2
SCHEMBL12629284 0.65 SLC1A3 (0.48) CYP1A2CYP3A4ADORA2AADORA1CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0353902-B1 SUBSTITUTED PHENYLTRIAZOLOPYRIMIDINE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-05-05 EP disclosed
US-5127936-A Substituted phenyltriazolopyrimidine herbicides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-07-07 US disclosed
WO-1990012012-A1 SUBSTITUTED PHENYLTRIAZOLOPYRIMIDINE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1990-10-18 WO disclosed
EP-0353902-A1 Substituted phenyltriazolopyrimidine herbicides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1990-02-07 EP disclosed