SCHEMBL9537543

SCHEMBL9537543

[CH](c1ccc(-c2ccccc2)cc1)c1nnn[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.34
CA1 P00915 1/20 0.34
MGLL Q99685 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
CHEK1 O14757 3/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
SIRT5 Q9NXA8 1/20 0.33
FGFR1 P11362 1/20 0.32
GP6 Q9HCN6 1/20 0.32
HDAC2 Q92769 1/20 0.32
DYRK3 O43781 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3656377 0.89 KMT2A (0.34) ALDH1A1CYP1A2L3MBTL1LMNANPC1
SCHEMBL9782419 0.78 PTGS2 (0.40) ALDH1A1CYP1A2CYP3A4CYP2C9TP53
SCHEMBL2457562 0.72 KMT2A (0.47) ALDH1A1CYP1A2LMNANPC1RAB9A
SCHEMBL2457565 0.72 KMT2A (0.47) ALDH1A1CYP1A2LMNANPC1RAB9A
SCHEMBL6505461 0.71 NR1H2 (0.41) ALDH1A1CYP1A2L3MBTL1LMNAFGFR1
SCHEMBL2839493 0.71 ALDH1A1 (0.56) ALDH1A1CYP1A2CYP3A4CYP2C9ATM
Bromide SCHEMBL27863912 0.69 NR1H2 (0.39) ALDH1A1CYP1A2L3MBTL1LMNAFGFR1
SCHEMBL5543150 0.69 CHRM5 (0.42) CYP1A2CYP2C9MAPTNPC1MEN1
SCHEMBL5540341 0.69 NFE2L2 (0.46) CYP1A2CYP3A4FGFR1NPC1RAB9A
SCHEMBL291507 0.69 ALDH1A1 (0.53) ALDH1A1CYP1A2CYP3A4TP53CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564960-A1 Imidazopyridines as angiotensin II antagonists MERCK PATENT GmbH (DE) 1993-10-13 EP disclosed