SCHEMBL9537613

SCHEMBL9537613

O=C1CCc2c(OCC3CO3)cccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
GLA P06280 1/20 0.50
ABCB1 P08183 2/20 0.47
TSHR P16473 2/20 0.45
TP53 P04637 1/20 0.45
CYP3A4 P08684 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HIF1A Q16665 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.44
TDP1 Q9NUW8 1/20 0.42
SLC6A4 P31645 2/20 0.42
ADRB2 P07550 1/20 0.42
ADRB1 P08588 1/20 0.42
HTR1A P08908 1/20 0.42
ADRB3 P13945 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
BRD4 O60885 2/20 0.41
MAPK14 Q16539 2/20 0.41
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8051434 0.93 MRGPRX4 (0.52) ALDH1A1GLAABCB1TSHRTP53
SCHEMBL9128670 0.93 MRGPRX4 (0.52) ALDH1A1GLAABCB1TSHRTP53
SCHEMBL11805028 0.92 ALDH1A1 (0.48) ALDH1A1GLAABCB1TSHRTP53
SCHEMBL11634077 0.82 HTR2A (0.60) ABCB1CYP3A4MRGPRX4SLC6A4ADRB2
SCHEMBL4814894 0.81 PKM (0.61) ALDH1A1ABCB1MRGPRX4LMNAPKM
SCHEMBL9197129 0.81 PARP1 (0.53) ALDH1A1GLATSHRTP53CYP3A4
SCHEMBL9447546 0.81 PARP1 (0.53) ALDH1A1GLATSHRTP53CYP3A4
SCHEMBL9447511 0.81 PARP1 (0.53) ALDH1A1GLATSHRTP53CYP3A4
SCHEMBL8057578 0.80 PARP1 (0.49) ALDH1A1GLATSHRTP53CYP3A4
SCHEMBL9311184 0.78 ALDH1A1 (0.56) ALDH1A1GLATSHRTP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5254595-A Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them ELF SANOFI (FR) 1993-10-19 US disclosed
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed
EP-0043971-B1 INDANONEOXYALKYLPIPERAZINE DERIVATIVES, THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME BASF Aktiengesellschaft (DE) 1984-12-19 EP disclosed
US-4435397-A ADRENERGIC BLOCKING AGENTS, 4-(3-ARYLOXY-2-HYDROXYPROPYL) SUBSTITUTED NIPPON SHINYAKU CO., LTD. (JP) 1984-03-06 US disclosed
EP-0043971-A1 Indanoneoxyalkylpiperazine derivatives, the preparation thereof and pharmaceutical compositions containing the same BASF Aktiengesellschaft (DE) 1982-01-20 EP disclosed
US-4109088-A ANTIDEPRESSANTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1978-08-22 US disclosed