SCHEMBL9538240

SCHEMBL9538240

O=C(NC1CCCCC1)N(S)C1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 8/20 0.50
NPC1 O15118 4/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
RAB9A P51151 3/20 0.50
MAPT P10636 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP3A4 P08684 1/20 0.50
EPHX2 P34913 1/20 0.50
ADRA2A P08913 1/20 0.45
PDE4A P27815 1/20 0.45
ADRA1A P35348 1/20 0.45
PKM P14618 1/20 0.44
MMP2 P08253 3/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
MMP8 P22894 1/20 0.42
MMP1 P03956 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11562576 0.85 EPHX2 (0.38) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL9547549 0.79 EPHX1 (0.54) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL27429391 0.78 EPHX1 (0.48) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL11634500 0.78 PKM (0.53) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL27736243 0.77 EPHX1 (0.47) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL679618 0.76 CCR5 (0.52) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL5705094 0.76 EPHX1 (0.50) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL25867965 0.76 EPHX1 (0.50) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL6684532 0.74 EPHX1 (0.48) EPHX1NPC1SMN1; SMN2RAB9AMAPT
SCHEMBL12506208 0.74 ADRA2A (0.56) EPHX1NPC1SMN1; SMN2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3979311-A MIXTURE OF AN ALKYNYL CYCLOALKANOL AND AN N,N'-DICYCLOALKYL-THIOUREA UNIVERSAL OIL PRODUCTS COMPANY (US) 1976-09-07 US claimed
US-3969260-A ALKYNYL CYCLOALKANOL, N,N'-DICYCLOALKYL THIOUREA, POLYAMINOMETHYLENEPHOSPHONATE UNIVERSAL OIL PRODUCTS COMPANY (US) 1976-07-13 US claimed
WO-1993002118-A1 A PROCESS FOR PREPARING ALKALI METAL SALTS OF POLYACRYLIC ACID BASED ON POLYSACCHARIDE TAECHANG MOOLSAN CO., LTD. (KR) 1993-02-04 WO disclosed
US-4159328-A INSECTICIDES, MITICIDES NIHON NOHYAKU CO., LTD. (JP) 1979-06-26 US disclosed
US-4061647-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DT) 1977-12-06 US disclosed
US-3984416-A Substituted quinoline-8-carboxamido ethyl benzene-sulfonyl N-cyclopentylmethyl urea HOECHST AKTIENGESELLSCHAFT (DT) 1976-10-05 US disclosed
US-3979311-A MIXTURE OF AN ALKYNYL CYCLOALKANOL AND AN N,N'-DICYCLOALKYL-THIOUREA UNIVERSAL OIL PRODUCTS COMPANY (US) 1976-09-07 US disclosed
US-3969260-A ALKYNYL CYCLOALKANOL, N,N'-DICYCLOALKYL THIOUREA, POLYAMINOMETHYLENEPHOSPHONATE UNIVERSAL OIL PRODUCTS COMPANY (US) 1976-07-13 US disclosed
US-3962244-A LOWERING OF BLOOD-SUGAR LEVELS HOECHST AKTIENGESELLSCHAFT (DT) 1976-06-08 US disclosed