SCHEMBL9538405

SCHEMBL9538405

CCCCCCn1c(C(=O)OCC)c(OC)c2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
HTT P42858 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.57
CNR2 P34972 5/20 0.55
KDM4E B2RXH2 3/20 0.54
LMNA P02545 1/20 0.54
MAPK1 P28482 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
PSEN1 P49768 1/20 0.52
PSEN2 P49810 1/20 0.52
APH1B Q8WW43 1/20 0.52
NCSTN Q92542 1/20 0.52
APH1A Q96BI3 1/20 0.52
PSENEN Q9NZ42 1/20 0.52
CNR1 P21554 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536349 1.00 ALDH1A1 (0.60) ALDH1A1HTTL3MBTL1CNR2KDM4E
SCHEMBL10762568 0.86 CCR2 (0.55) KDM4EMAPK1NPSR1PSEN1PSEN2
SCHEMBL10758013 0.86 CCR2 (0.55) KDM4EMAPK1NPSR1PSEN1PSEN2
SCHEMBL8358463 0.85 ALDH1A1 (0.76) ALDH1A1HTTL3MBTL1CNR2KDM4E
SCHEMBL9259706 0.85 ALDH1A1 (0.76) ALDH1A1HTTL3MBTL1CNR2KDM4E
SCHEMBL9868002 0.81 ALDH1A1 (0.54) ALDH1A1L3MBTL1KDM4ENPSR1
SCHEMBL9538311 0.81 CCR2 (0.60) ALDH1A1KDM4ELMNAMAPK1
SCHEMBL31383501 0.79 KDM4E (0.60) ALDH1A1HTTL3MBTL1CNR2KDM4E
SCHEMBL11185256 0.78 KDM4E (0.46) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL5797851 0.77 CNR2 (0.73) ALDH1A1CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0186367-B1 ACIDIC INDOLE COMPOUNDS AND THEIR USE AS ANTIALLERGY AGENTS WARNER-LAMBERT COMPANY (US) 1993-03-03 EP disclosed
US-4675332-A Acidic tetrazolyl substituted indole compounds and their use as antiallergy agents WARNER-LAMBERT COMPANY (US) 1987-06-23 US disclosed
EP-0186367-A2 Acidic indole compounds and their use as antiallergy agents WARNER-LAMBERT COMPANY (US) 1986-07-02 EP disclosed