SCHEMBL9538969

SCHEMBL9538969

FC(F)(F)c1ccc2c(C=P(c3ccccc3)(c3ccccc3)c3ccccc3)cc(C(F)(F)F)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.39
ESR1 P03372 1/20 0.38
DGAT1 O75907 1/20 0.38
KCNH2 Q12809 1/20 0.38
NT5E P21589 3/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
DHODH Q02127 1/20 0.36
BACE1 P56817 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CCNE2 O96020 1/20 0.35
CCNA2 P20248 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
F7 P08709 1/20 0.35
F3 P13726 1/20 0.35
C1R P00736 1/20 0.34
CTSD P07339 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538889 0.75 NPBWR1 (0.40) NPBWR1ESR1DGAT1KCNH2DHODH
SCHEMBL9541219 0.74 ESR1 (0.41) ESR1KCNH2ADORA2AADORA1BACE1
SCHEMBL9538666 0.74 NPBWR1 (0.39) NPBWR1DGAT1KCNH2BACE1
SCHEMBL9735498 0.71 TOP1 (0.35) ESR1NT5EADORA2AADORA1KDM4E
SCHEMBL19209593 0.70 GAA (0.52) KDM4EC1RABCG2TLR7
SCHEMBL31327779 0.70 NT5E (0.68) NPBWR1DGAT1KCNH2NT5EADORA2A
SCHEMBL2709353 0.70 NT5E (0.68) NPBWR1DGAT1KCNH2NT5EADORA2A
SCHEMBL3826784 0.70 NT5E (0.54) NT5EBACE1KDM4EF7F3
SCHEMBL3828474 0.68 BACE1 (0.45) NT5EBACE1KDM4EF7F3
SCHEMBL11133397 0.68 KDM4E (0.49) DGAT1KCNH2NT5EADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed