SCHEMBL9538889

SCHEMBL9538889

FC(F)(F)c1ccc(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.40
DGAT1 O75907 1/20 0.38
KCNH2 Q12809 1/20 0.38
CES2 O00748 2/20 0.38
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
KIF11 P52732 2/20 0.36
BACE1 P56817 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
POLQ O75417 1/20 0.35
TRPV6 Q9H1D0 1/20 0.35
CBFB Q13951 1/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
AVPR2 P30518 1/20 0.34
GPR27 Q9NS67 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538666 0.83 NPBWR1 (0.39) NPBWR1DGAT1KCNH2ALDH1A1TSHR
SCHEMBL9538969 0.75 NPBWR1 (0.39) NPBWR1DGAT1KCNH2BACE1CBFB
SCHEMBL5255552 0.75 CES2 (0.41) NPBWR1DGAT1KCNH2CES2ALDH1A1
SCHEMBL9539528 0.74 ALDH1A1 (0.48) ALDH1A1TSHRKIF11BACE1TRPV6
SCHEMBL9540307 0.73 FBP1 (0.47) ALDH1A1TSHRMEN1MAPTKMT2A
SCHEMBL9541838 0.73 IDO1 (0.44) ALDH1A1TSHRKIF11KDM4EMEN1
SCHEMBL4416163 0.71 CES2 (0.47) NPBWR1CES2KIF11BACE1POLQ
SCHEMBL9996772 0.70 CES2 (0.46) NPBWR1CES2TSHRBACE1KDM4E
SCHEMBL4076004 0.70 CES2 (0.46) NPBWR1CES2TSHRBACE1KDM4E
SCHEMBL472401 0.70 CES2 (0.50) CES2KIF11BACE1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed