SCHEMBL9539338

SCHEMBL9539338

O=C(OCc1ccccc1)Oc1nnc(O)c2[nH]cnc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 2/20 0.38
CYP1A2 P05177 1/20 0.38
CDK1 P06493 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CCNB1 P14635 1/20 0.38
MGMT P16455 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540456 0.79 ALOX5 (0.36) HSD17B10LMNACDK1CCNB1MGMT
SCHEMBL9540433 0.77 LMNA (0.43) L3MBTL1LMNACYP1A2CDK1CYP3A4
SCHEMBL10359891 0.69 KMT2A (0.52) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL9542967 0.67 CSNK2A2 (0.34) KMT2AMEN1MGMTTSHR
SCHEMBL37382 0.66 ALDH1A1 (0.68) KMT2AL3MBTL1LMNATSHRALDH1A1
SCHEMBL22162939 0.65 KMT2A (0.54) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL697595 0.65 KMT2A (0.60) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL22882716 0.65 ALDH1A1 (0.57) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL6943583 0.64 KMT2A (0.44) KMT2AMEN1HTTGFERHSD17B10
SCHEMBL1927968 0.64 LMNA (0.59) KMT2AMEN1HTTGFERHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003033-A1 CARBONATE-SUBSTITUTED IMIDAZO[4,5-d] PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G. D. SEARLE & CO. (US) 1993-02-18 WO claimed
WO-1993003033-A1 CARBONATE-SUBSTITUTED IMIDAZO[4,5-d] PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G. D. SEARLE & CO. (US) 1993-02-18 WO disclosed