SCHEMBL95394

SCHEMBL95394

Nc1nc(O)nc2[nH]ncc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 3/20 0.52
RET P07949 1/20 0.52
PI4KA P42356 1/20 0.52
LRRK2 Q5S007 1/20 0.52
PI4K2B Q8TCG2 1/20 0.52
PI4K2A Q9BTU6 1/20 0.52
PI4KB Q9UBF8 1/20 0.52
ADORA2A P29274 3/20 0.37
ADORA1 P30542 2/20 0.37
CDK2 P24941 2/20 0.37
GRK2 P25098 1/20 0.35
CHEK1 O14757 2/20 0.35
PDPK1 O15530 1/20 0.35
AURKA O14965 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 2/20 0.33
RAB9A P51151 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13829440 0.80 RET (0.52) XDHRETPI4KALRRK2PI4K2B
Oxypurinol SCHEMBL49280 0.79 SMN1; SMN2 (0.38) XDHRETPI4KALRRK2PI4K2B
SCHEMBL1014920 0.79 XDH (0.55) XDHRETPI4KALRRK2PI4K2B
SCHEMBL29487078 0.79 XDH (0.55) XDHRETPI4KALRRK2PI4K2B
Oxypurinol SCHEMBL5799552 0.78 SMN1; SMN2 (0.37) XDHRETPI4KALRRK2PI4K2B
Oxypurinol SCHEMBL8905835 0.78 SMN1; SMN2 (0.37) XDHRETPI4KALRRK2PI4K2B
Oxypurinol SCHEMBL8905886 0.78 SMN1; SMN2 (0.37) XDHRETPI4KALRRK2PI4K2B
Oxypurinol SCHEMBL8905476 0.78 SMN1; SMN2 (0.37) XDHRETPI4KALRRK2PI4K2B
Benzene SCHEMBL25427466 0.76 RET (0.52) XDHRETPI4KALRRK2PI4K2B
SCHEMBL8141335 0.76 XDH (0.34) XDHRETPI4KALRRK2PI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 101 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4560315-A2 HYBRIDIZING ALL-LNA OLIGONUCLEOTIDES F. Hoffmann-La Roche AG (CH) 2025-05-28 EP claimed
EP-3980554-B1 HYBRIDIZING ALL-LNA OLIGONUCLEOTIDES HOFFMANN LA ROCHE (CH) 2025-03-26 EP claimed
US-20220195497-A1 HYBRIDIZING all-LNA OLIGONUCLEOTIDES ROCHE DIAGNOSTICS OPERATIONS, INC. 2022-06-23 US claimed
EP-3980554-A1 HYBRIDIZING ALL-LNA OLIGONUCLEOTIDES F. Hoffmann-La Roche AG (CH) 2022-04-13 EP claimed
CN-113939599-A Hybrid all-LNA oligonucleotides 豪夫迈·罗氏有限公司 2022-01-14 CN claimed
WO-2020245377-A1 HYBRIDIZING ALL-LNA OLIGONUCLEOTIDES F. HOFFMANN-LA ROCHE AG (CH) 2020-12-10 WO claimed
US-7829596-B2 Methods of treatment IMPERIAL INNOVATIONS LIMITED (GB) 2010-11-09 US claimed
US-20090023639-A1 Methods of Treatment IMPERIAL INNOVATIONS LIMITED (GB) 2009-01-22 US claimed
EP-0759298-B1 Use of 4-amino-6-hydroxypyrazolo[3,4-d]pyrimidine for the manufacture of an antihypertensive agent MAEDA HIROSHI DR (JP) 2003-11-05 EP claimed
EP-0881875-A4 COMPOSITIONS AND METHODS FOR CONTROLLING PEST INSECTS VIRGINIA TECH INTELL PROP (US) 2002-03-06 EP claimed
WO-2000021509-A2 METHODS OF TREATMENT IMPERIAL COLLEGE INNOVATIONS LIMITED (GB) 2000-04-20 WO claimed
US-6037344-A COMPRISING A PURINE SELECTED FROM THE GROUP CONSISTING OF XANTHINE, HYPOXANTHINE, GUANINE AND MIXTURES THEREOF, AND A XANTHINE OXIDASE INHIBITOR SELECTED FROM THE GROUP CONSISTING OF ALLOPURINOL, OXYPURINOL, MERCAPTO-ALLOPURINOL, VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2000-03-14 US claimed
EP-0881875-A1 COMPOSITIONS AND METHODS FOR CONTROLLING PEST INSECTS VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 1998-12-09 EP claimed
WO-1997028686-A1 COMPOSITIONS AND METHODS FOR CONTROLLING PEST INSECTS VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 1997-08-14 WO claimed
EP-0759298-A2 Pyrazolopyrimidine derivates as antihypertensive agents Maeda, Hiroshi, Dr. (JP) 1997-02-26 EP claimed
EP-0515379-A4 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INC (US) 1994-09-14 EP claimed
EP-0515379-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1992-12-02 EP claimed
US-5094740-A TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED, INC. (US) 1992-03-10 US claimed
WO-1991012275-A1 TWO-DIMENSIONAL ELECTROPHORETIC SEPARATION OF CARBOHYDRATES GLYCOMED INCORPORATED (US) 1991-08-22 WO claimed
WO-1991012276-A1 ELECTRO-BLOTTING OF ELECTROPHORETICALLY RESOLVED FLUORESCENT-LABELED SACCHARIDES AND DETECTION OF ACTIVE STRUCTURES WITH PROTEIN PROBES GLYCOMED INCORPORATED (US) 1991-08-22 WO claimed