SCHEMBL9539740

SCHEMBL9539740

Cc1ccc(-c2ccc(COCCN(O)C(N)=O)s2)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.39
HSD17B1 P14061 5/20 0.39
HSD17B2 P37059 5/20 0.39
ESRRG P62508 2/20 0.36
ALOX5 P09917 6/20 0.34
ACKR3 P25106 1/20 0.34
RORC P51449 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9585017 0.88 IKBKB (0.46) MMP2ESRRGALOX5ESR1
SCHEMBL9584912 0.87 CYP2E1 (0.45) MMP2ALOX5CYP2C9CYP2C19
SCHEMBL9538854 0.83 IKBKB (0.42) MMP2ALOX5CYP2C9CYP2C19
SCHEMBL9539825 0.83 ALOX5 (0.39) MMP2ALOX5
SCHEMBL9585668 0.77 ALOX5 (0.49) MMP2ALOX5CYP1A2CYP2C9HPGD
SCHEMBL9583758 0.74 MMP2 (0.33) MMP2ALOX5
SCHEMBL9584641 0.73 MMP2 (0.37) MMP2ALOX5
SCHEMBL9584629 0.72 MMP2 (0.34) MMP2ALOX5
SCHEMBL9584273 0.71 ALOX5 (0.42) MMP2HSD17B1HSD17B2ALOX5
SCHEMBL9375297 0.70 CYP2E1 (0.50) ALOX5CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003719-A1 ARYLALKYLETHER AND ARYLALKYLTHIOETHER INHIBITORS OF LIPOXYGENASE ENZYME ACTIVITY ABBOTT LABORATORIES (US) 1993-03-04 WO claimed
US-5183818-A Also for inhibiting leukotriene biosynthesis ABBOTT LABORATORIES (US) 1993-02-02 US disclosed