SCHEMBL9540065

SCHEMBL9540065

C=CCn1c(CCCCC)c2ccccc2nc1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.51
ATM Q13315 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
LMNA P02545 3/20 0.46
TSHR P16473 1/20 0.46
TP53 P04637 2/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
ALDH1A1 P00352 7/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
PARP1 P09874 1/20 0.41
MAPK1 P28482 1/20 0.41
GAA P10253 3/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.40
TLR8 Q9NR97 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3636224 0.78 RORA (0.44) TDP1LMNATSHRTP53ALDH1A1
SCHEMBL20274635 0.72 LMNA (0.43) TDP1ATMLMNAALDH1A1L3MBTL1
SCHEMBL6527375 0.71 TP53 (0.66) LMNATSHRTP53MAPK1GAA
SCHEMBL6027390 0.70 TDP1 (0.60) TDP1SMN1; SMN2LMNATSHRALDH1A1
SCHEMBL5553536 0.69 PDE4B (0.38) TDP1ATMSMN1; SMN2LMNATSHR
SCHEMBL2731836 0.69 TDP1 (0.62) TDP1SMN1; SMN2LMNATSHRALDH1A1
SCHEMBL11498915 0.68 TSHR (0.59) TDP1ATMSMN1; SMN2LMNATSHR
SCHEMBL11053715 0.67 ALDH1A1 (0.53) LMNATP53ALDH1A1MAPTPOLB
SCHEMBL4925728 0.67 KMT2A (0.46) TDP1SMN1; SMN2LMNATP53ALDH1A1
SCHEMBL6279426 0.67 HCAR2 (0.39) LMNATP53ALDH1A1L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed