SCHEMBL9540446

SCHEMBL9540446

O=C(Oc1nnc(O)c2nc[nH]c12)OC1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CDK1 P06493 3/20 0.32
CDK2 P24941 3/20 0.32
CCNB2 O95067 2/20 0.32
CCNB1 P14635 2/20 0.32
CCNA2 P20248 2/20 0.32
CCNA1 P78396 2/20 0.32
CCNB3 Q8WWL7 2/20 0.32
CYP19A1 P11511 3/20 0.32
EPHX1 P07099 2/20 0.31
MMP9 P14780 2/20 0.31
MMP12 P39900 2/20 0.31
MMP1 P03956 1/20 0.31
MAPK3 P27361 1/20 0.30
CLK1 P49759 1/20 0.30
CDK5 Q00535 1/20 0.30
PIN1 Q13526 1/20 0.30
MAP3K5 Q99683 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543043 0.93 ALDH1A1 (0.38) ALDH1A1HPGDHSD17B10CDK1CDK2
SCHEMBL9540186 0.64 LMNA (0.46) ALDH1A1HPGDCDK1CDK2CCNB1
SCHEMBL28445719 0.62 STS (0.43) ALDH1A1HSD17B10CYP19A1EPHX1MMP9
SCHEMBL31643443 0.61 MMP9 (0.41) ALDH1A1CYP19A1EPHX1MMP9MMP12
SCHEMBL11589654 0.61 EPHX1 (0.60) ALDH1A1EPHX1SMN1; SMN2
SCHEMBL13387598 0.61 EPHX1 (0.60) ALDH1A1EPHX1SMN1; SMN2
SCHEMBL8426647 0.61 EPHX1 (0.60) ALDH1A1EPHX1SMN1; SMN2
SCHEMBL8991654 0.61 EPHX1 (0.60) ALDH1A1EPHX1SMN1; SMN2
SCHEMBL984315 0.61 EPHX1 (0.60) ALDH1A1EPHX1SMN1; SMN2
SCHEMBL37472 0.61 EPHX1 (0.60) ALDH1A1EPHX1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003033-A1 CARBONATE-SUBSTITUTED IMIDAZO[4,5-d] PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G. D. SEARLE & CO. (US) 1993-02-18 WO claimed