SCHEMBL9540887

SCHEMBL9540887

COc1ccc2c(c1)C1(C)CCN(CC=C(C)C)C1N2C

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 12/20 0.58
BCHE P06276 11/20 0.58
KDM4E B2RXH2 2/20 0.47
CYP2D6 P10635 2/20 0.47
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
KMT2A Q03164 1/20 0.47
HIF1A Q16665 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
PTGS1 P23219 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
BLM P54132 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9537459 0.99 ACHE (0.57) ACHEBCHEKDM4ECYP2D6MEN1
SCHEMBL8827811 0.87 ACHE (0.71) ACHEBCHEKDM4ECYP2D6MEN1
SCHEMBL8827817 0.87 ACHE (0.71) ACHEBCHEKDM4ECYP2D6MEN1
SCHEMBL9537558 0.87 ACHE (0.71) ACHEBCHEKDM4ECYP2D6MEN1
Hydrochloric Acid SCHEMBL9540534 0.86 ACHE (0.70) ACHEBCHEKDM4ECYP2D6MEN1
SCHEMBL9537601 0.82 SIGMAR1 (0.45) ACHEBCHEOPRM1OPRK1
SCHEMBL9006729 0.81 ACHE (0.51) ACHEBCHEKDM4ECYP2D6MEN1
SCHEMBL8863165 0.81 ACHE (0.51) ACHEBCHEKDM4ECYP2D6MEN1
SCHEMBL8863164 0.81 ACHE (0.51) ACHEBCHEKDM4ECYP2D6MEN1
Hydrochloric Acid SCHEMBL9537532 0.80 ACHE (0.50) ACHEBCHEKDM4ECYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5187165-A Eseroline derivatives; cholinergic agents; antidepressants HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-02-16 US disclosed