SCHEMBL9540919

SCHEMBL9540919

CC(C)Oc1ccccc1N1CCN(CCc2cccc(C(=O)N3CCCCC3)c2)CC1

nearest known ligand 0.82

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 3/20 0.82
ADRA1A P35348 3/20 0.82
ADRA1B P35368 3/20 0.82
HTR1A P08908 1/20 0.82
DRD2 P14416 1/20 0.82
HTR1B P28222 1/20 0.82
DRD3 P35462 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7648376 0.96 ADRA1D (0.77) ADRA1DADRA1AADRA1BHTR1ADRD2
Mazapertine SCHEMBL636631 0.90 HTR1A (1.00) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL13533242 0.90 HTR1A (1.00) ADRA1DADRA1AADRA1BHTR1ADRD2
Mazapertine SCHEMBL7643633 0.90 HTR1A (0.98) ADRA1DADRA1AADRA1BHTR1ADRD2
Hydrochloric Acid SCHEMBL7644692 0.90 HTR1A (0.98) ADRA1DADRA1AADRA1BHTR1ADRD2
Oxalic Acid SCHEMBL7647400 0.87 ADRA1D (0.67) ADRA1DADRA1AADRA1BHTR1ADRD2
Mazapertine SCHEMBL6013382 0.86 HTR1A (0.91) ADRA1DADRA1AADRA1BHTR1ADRD2
Mazapertine SCHEMBL120658 0.86 HTR1A (0.91) ADRA1DADRA1AADRA1BHTR1ADRD2
Mazapertine SCHEMBL1649526 0.86 HTR1A (0.91) ADRA1DADRA1AADRA1BHTR1ADRD2
Bromide SCHEMBL7647385 0.82 ADRA1D (0.64) ADRA1DADRA1AADRA1BHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563345-A1 NOVEL 4-ARYLPIPERAZINES AND 4-ARYLPIPERIDINES MCNEILAB, INC. (US) 1993-10-06 EP disclosed
WO-1993004682-A1 NOVEL 4-ARYLPIPERAZINES AND 4-ARYLPIPERIDINES MCNEILAB, INC. (US) 1993-03-18 WO disclosed