SCHEMBL9541551

SCHEMBL9541551

CC(=O)Nc1nc(CC(C)(OC(N)=O)C(=O)NCCc2ccccc2)cs1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 12/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAOB P27338 1/20 0.46
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
CASP3 P42574 1/20 0.42
HTT P42858 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7672023 0.82 AOC3 (0.47) AOC3NPC1RAB9ASMN1; SMN2MAOB
SCHEMBL9700657 0.78 MMP8 (0.46) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9541051 0.77 MMP8 (0.44) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9539323 0.75 MMP8 (0.51) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL9539180 0.75 MMP8 (0.44) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL8430108 0.74 AOC3 (0.76) AOC3NPC1RAB9ASMN1; SMN2MAOB
SCHEMBL9541636 0.74 MMP8 (0.49) NPC1RAB9ASMN1; SMN2POLBALDH1A1
SCHEMBL9538003 0.74 MMP8 (0.46) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL9538757 0.74 MTNR1A (0.50) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL4890202 0.73 AOC3 (0.73) AOC3SMN1; SMN2MAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed