Bromide

Bromide

SCHEMBL9542002

Br.Cc1c(CBr)cnc2nc(N)nc(N)c12

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.63
SLC2A1 P11166 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319768 0.98 DHFR (0.64) DHFRSLC2A1
SCHEMBL9068396 0.83 DHFR (0.60) DHFRSLC2A1
SCHEMBL8322799 0.80 DHFR (0.51) DHFRSLC2A1
SCHEMBL10465515 0.78 DHFR (0.74) DHFRSLC2A1
SCHEMBL5462527 0.78 DHFR (0.58) DHFRSLC2A1
SCHEMBL8322368 0.78 DHFR (0.46) DHFRSLC2A1
SCHEMBL27188510 0.76 DHFR (0.52) DHFRSLC2A1
SCHEMBL30092875 0.76 DHFR (0.52) DHFRSLC2A1
SCHEMBL9549873 0.74 DHFR (0.48) DHFRSLC2A1
SCHEMBL10052933 0.74 DHFR (0.82) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4725687-A ANTITUMOR AGENTS; SIDE EFFECT REDUCTION; POTENCY SOUTHERN RESEARCH INSTITUTE (US) 1988-02-16 US claimed
WO-1993013102-A1 DEAZAAMINOPTERINS SOUTHERN RESEARCH INSTITUTE (US) 1993-07-08 WO disclosed
US-5077404-A Cyclized 5,10-dideazaaminopterin compounds SRI INTERNATIONAL 1991-12-31 US disclosed