SCHEMBL9542849

SCHEMBL9542849

CC(C)(C)OC(=O)NCc1cccc(C2CCN(Cc3ccccc3)C2)c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.49
CHRM4 P08173 4/20 0.49
DRD2 P14416 3/20 0.48
NPFFR1 Q9GZQ6 1/20 0.46
NPFFR2 Q9Y5X5 1/20 0.46
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
BCHE P06276 1/20 0.44
DRD4 P21917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27679079 0.87 CHRM4 (0.43) ROCK2CHRM4DRD2DRD4
SCHEMBL7981628 0.85 CHRM4 (0.53) CHRM4DRD2NPFFR1NPFFR2KMT2A
SCHEMBL3509882 0.83 BRD4 (0.48) ROCK2L3MBTL1
SCHEMBL30531024 0.83 BRD4 (0.48) ROCK2L3MBTL1
SCHEMBL15866724 0.83 ACHE (0.49)
SCHEMBL13830591 0.82 QDPR (0.45) ROCK2CHRM4
SCHEMBL25358558 0.81 GLS (0.48) ROCK2KMT2AL3MBTL1
SCHEMBL30531063 0.81 GLS (0.48) ROCK2KMT2AL3MBTL1
SCHEMBL25048390 0.81 BRD4 (0.47) ROCK2KMT2AL3MBTL1
SCHEMBL7766536 0.81 DRD4 (0.69) DRD2KMT2ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993016077-A1 7-SUBSTITUTED QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1993-08-19 WO disclosed