SCHEMBL9543189

SCHEMBL9543189

C=C(c1nc2ccccc2n1Cc1ccc(F)cc1)C1CCN(C)CC1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 13/20 0.57
TACR2 P21452 1/20 0.57
TACR1 P25103 1/20 0.57
CYP2D6 P10635 11/20 0.56
KCNH2 Q12809 7/20 0.56
CHRM1 P11229 5/20 0.56
TP53 P04637 1/20 0.51
RAB9A P51151 1/20 0.50
SSTR5 P35346 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541656 0.89 HRH1 (0.61) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9544433 0.88 HRH1 (0.58) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9264751 0.87 HRH1 (0.72) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9259609 0.77 HRH1 (0.67) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9258632 0.77 HRH1 (0.56) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL10529762 0.76 SSTR5 (0.78) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9196229 0.76 HRH1 (0.66) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9697152 0.76 HRH1 (0.73) HRH1TACR2TACR1CYP2D6KCNH2
SCHEMBL9543194 0.74 HRH1 (0.56) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL9259670 0.74 HRH1 (0.69) HRH1TACR2TACR1CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014083-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED BENZIMIDAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-07-22 WO disclosed