SCHEMBL9543252

SCHEMBL9543252

COC(=O)CCNC(=O)[C@@H]1Cc2ccccc2N1C(=O)[C@H](CCc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 5/20 0.51
CTSK P43235 2/20 0.47
CTSS P25774 1/20 0.47
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
XIAP P98170 1/20 0.44
ACE P12821 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543250 0.86 ACE (0.51) CXCR3CTSKCTSSXIAPACE
SCHEMBL9544867 0.85 CTSK (0.48) CTSKCTSSACE
SCHEMBL9545294 0.82 CCKBR (0.44)
SCHEMBL9542638 0.79 KDM4E (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9542646 0.79 KDM4E (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9544975 0.79 CTSK (0.51) CTSKCTSSACE
SCHEMBL9544256 0.79 CTSK (0.51) CTSKCTSSACE
SCHEMBL5564454 0.77 KDM4E (0.52) CXCR3KDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9543558 0.76 ACE (0.52) CTSKACE
SCHEMBL9543550 0.76 ACE (0.52) CTSKACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993020099-A2 CCK AND/OR GASTRIN RECEPTOR LIGANDS FERRING B.V. (NL) 1993-10-14 WO disclosed