SCHEMBL9543804

SCHEMBL9543804

COc1ccc(C(=O)Cl)c(OC(=O)C(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
NPC1 O15118 2/20 0.45
KMT2A Q03164 3/20 0.43
MAPT P10636 4/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
ELANE P08246 1/20 0.42
CYP3A4 P08684 1/20 0.41
MAPK1 P28482 1/20 0.41
ABCG2 Q9UNQ0 3/20 0.41
RAD52 P43351 1/20 0.41
TNFRSF1A P19438 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805920 0.83 KDM4E (0.58) NPC1KMT2AMAPTALDH1A1HPGD
SCHEMBL15548524 0.82 ALOX15 (0.57) TP53NPC1KMT2AMAPTALDH1A1
SCHEMBL220681 0.82 NPC1 (0.64) TP53NPC1KMT2AMAPTALDH1A1
SCHEMBL20204164 0.81 TP53 (0.48) TP53NPC1KMT2AMAPTALDH1A1
SCHEMBL9543811 0.79 HDAC3 (0.44) TP53NPC1KMT2AMAPTALDH1A1
SCHEMBL11184716 0.78 TAS1R3 (0.46) KMT2AMAPTALDH1A1MEN1ELANE
SCHEMBL27580216 0.76 KDM4E (0.58) NPC1KMT2AMAPTALDH1A1HPGD
SCHEMBL11252289 0.76 KDM4E (0.55) TP53NPC1MAPTHPGDRAB9A
SCHEMBL1914036 0.76 KDM4E (0.46) KMT2AMAPTALDH1A1HPGDMEN1
SCHEMBL14744132 0.76 KDM4E (0.72) TP53NPC1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed