SCHEMBL9543816

SCHEMBL9543816

COC(=O)C(C)c1cc(OC)ccc1C(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PTGS2 P35354 3/20 0.41
PTGS1 P23219 2/20 0.41
AKR1C3 P42330 2/20 0.41
AKR1C2 P52895 2/20 0.41
TSHR P16473 2/20 0.41
CDC42 P60953 1/20 0.41
RAC1 P63000 1/20 0.41
CYP1A2 P05177 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.41
HTT P42858 3/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL837247 0.81 TDP1 (0.44) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL4981399 0.80 CYP2D6 (0.58) RAB9AALDH1A1MAPK1TSHRCYP1A2
SCHEMBL31207283 0.78 HPGD (0.48) NPC1RAB9ACYP3A4HPGDTDP1
SCHEMBL1536363 0.75 HTT (0.58) NPC1RAB9ACYP3A4ALDH1A1HPGD
SCHEMBL1922871 0.75 PTGS2 (0.48) RAB9ATDP1L3MBTL1PTGS2PTGS1
SCHEMBL31207244 0.75 NPC1 (0.45) TP53NPC1RAB9ACYP3A4ALDH1A1
SCHEMBL11197823 0.75 NPC1 (0.55) NPC1RAB9ACYP3A4ALDH1A1HPGD
SCHEMBL9543804 0.73 TP53 (0.46) TP53NPC1RAB9ACYP3A4ALDH1A1
SCHEMBL9541390 0.72 KDM4E (0.58) NPC1RAB9ACYP3A4ALDH1A1HPGD
SCHEMBL20204164 0.72 TP53 (0.48) TP53NPC1RAB9ACYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed