SCHEMBL9544220

SCHEMBL9544220

Cn1ccc2cc(N(C(N)=O)c3cccc4ncccc34)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.47
HTR2C P28335 2/20 0.47
NTSR1 P30989 1/20 0.40
GRK5 P34947 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM1A O60341 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3R1 P27986 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
EGFR P00533 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098140 0.85 HTR2B (0.42) HTR2BHTR2CNTSR1GRK5MEN1
SCHEMBL9545059 0.85 GRM4 (0.39) HTR2BHTR2CGRK5MEN1KMT2A
SCHEMBL9542979 0.85 GRK5 (0.47) HTR2BHTR2CGRK5MEN1KMT2A
Hydrochloric Acid SCHEMBL5964207 0.84 HTR2C (0.42) HTR2BHTR2CNTSR1GRK5MEN1
SCHEMBL27407225 0.84 HTR2B (0.39) HTR2BHTR2CGRK5MEN1KMT2A
Hydrochloric Acid SCHEMBL27407226 0.83 HTR2C (0.40) HTR2BHTR2CGRK5MEN1KMT2A
SCHEMBL7378778 0.82 KDM1A (0.41) HTR2BHTR2CMEN1KMT2ATP53
SCHEMBL9544511 0.81 MAPT (0.42) HTR2BHTR2CNTSR1MEN1KMT2A
Hydrochloric Acid SCHEMBL9372300 0.81 KDM1A (0.41) HTR2BHTR2CMEN1KMT2ATP53
Hydrochloric Acid SCHEMBL9544563 0.78 HTR2C (0.41) HTR2BHTR2CNTSR1GRK5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018028-A1 INDOLE DERIVATIVES AS 5HT1C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-09-16 WO claimed
WO-1993018028-A1 INDOLE DERIVATIVES AS 5HT1C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-09-16 WO disclosed