SCHEMBL7378778

SCHEMBL7378778

Cc1cc(N(C(N)=O)c2ccc3c(ccn3C)c2)c2ccccc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
HSD11B1 P28845 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP1A2 P05177 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9372300 0.99 KDM1A (0.41) KDM1AHTR2CHTR2BHSD11B1SMN1; SMN2
SCHEMBL9544220 0.82 HTR2B (0.47) KDM1AHTR2CHTR2BMEN1KMT2A
SCHEMBL23037546 0.82 KDM1A (0.47) KDM1AHTR2CHTR2BHSD11B1CYP1A2
SCHEMBL6592538 0.81 NCF1 (0.47) SMN1; SMN2MEN1KMT2ACYP1A2NPC1
SCHEMBL6589107 0.81 CYP1A2 (0.44) SMN1; SMN2MEN1KMT2ACYP1A2NPC1
SCHEMBL6185025 0.80 NCF1 (0.51) SMN1; SMN2MEN1KMT2ACYP1A2NPC1
SCHEMBL9375448 0.80 CYP11B1 (0.43) KDM1AHTR2CHTR2BMEN1KMT2A
SCHEMBL7381173 0.78 GRM2 (0.44) SMN1; SMN2MEN1KMT2ACYP1A2LMNA
SCHEMBL6593276 0.78 CYP1A2 (0.41) SMN1; SMN2MEN1KMT2ACYP1A2NPC1
SCHEMBL9190817 0.78 ALDH1A1 (0.43) KDM1ASMN1; SMN2MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150977-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2001-11-07 EP claimed
WO-2000047577-A1 PHENYL UREA AND PHENYL THIOUREA DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2000-08-17 WO claimed
WO-1993018028-A1 INDOLE DERIVATIVES AS 5HT1C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-09-16 WO claimed