SCHEMBL9545059

SCHEMBL9545059

Cn1ccc2cc(N(C(N)=O)c3cccc4cccnc34)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.39
HTR2B P41595 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C19 P33261 1/20 0.39
RECQL P46063 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PARP1 P09874 2/20 0.39
HTR2C P28335 2/20 0.38
GRK5 P34947 1/20 0.38
PIK3CD O00329 1/20 0.37
PIK3R1 P27986 1/20 0.37
NSD2 O96028 1/20 0.36
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098140 0.87 HTR2B (0.42) GRM4HTR2BKDM4EMEN1TP53
Hydrochloric Acid SCHEMBL5964207 0.86 HTR2C (0.42) GRM4HTR2BKDM4EMEN1TP53
SCHEMBL27407225 0.86 HTR2B (0.39) GRM4HTR2BKDM4EMEN1TP53
SCHEMBL9544220 0.85 HTR2B (0.47) GRM4HTR2BKDM4EMEN1TP53
Hydrochloric Acid SCHEMBL27407226 0.85 HTR2C (0.40) GRM4HTR2BKDM4EMEN1TP53
SCHEMBL9542979 0.84 GRK5 (0.47) HTR2BKDM4EMEN1TP53CYP1A2
SCHEMBL9544511 0.81 MAPT (0.42) HTR2BKDM4EMEN1TP53CYP1A2
SCHEMBL9544345 0.80 HTR2B (0.40) GRM4HTR2BKDM4EMEN1TP53
SCHEMBL27469254 0.80 HTR2B (0.40) HTR2BKDM4EMEN1TP53CYP1A2
Hydrochloric Acid SCHEMBL9544563 0.78 HTR2C (0.41) HTR2BKDM4EMEN1TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018028-A1 INDOLE DERIVATIVES AS 5HT1C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-09-16 WO claimed