SCHEMBL954853

SCHEMBL954853

Brc1cccc(P(c2cccc(Br)n2)c2cccc(Br)n2)n1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ALOX5 P09917 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8160391 0.84 KDM4E (0.50) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL1219299 0.84 KDM4E (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3973 0.76
SCHEMBL29539234 0.69 CCR1 (0.46) HTR7HTR1ADRD2HTR2AGRIN2D
SCHEMBL229994 0.69 CCR1 (0.46) HTR7HTR1ADRD2HTR2AGRIN2D
SCHEMBL8155898 0.69 BTK (0.40) ALDH1A1HPGDALOX5GRM5
SCHEMBL8155129 0.68 TSHR (0.44) ALDH1A1HPGDGRM5
SCHEMBL955795 0.68 CCR1 (0.52) GRIN2BALDH1A1HPGDGRM5
SCHEMBL31354842 0.67 CCR1 (0.46) HTR7HTR1ADRD2HTR2AGRIN2D
SCHEMBL700152 0.67 CCR1 (0.46) HTR7HTR1ADRD2HTR2AGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861140-A Tripodal paramagnetic contrast agents for MR imaging HOECHST CELANESE CORP. (US) 1999-01-19 US claimed
US-5861138-A Ligands for MRI contrast agent HOECHST CELANESE CORP. (US) 1999-01-19 US claimed
WO-1998022148-A1 MRI CONTRAST AGENTS AND LIGANDS WASHINGTON UNIVERSITY (US) 1998-05-28 WO claimed
US-8617723-B2 Metal complexes MERCK PATENT GMBH (DE) 2013-12-31 US disclosed
WO-2011066898-A1 ELECTRONIC DEVICE CONTAINING METAL COMPLEXES MERCK PATENT GMBH (DE) 2011-06-09 WO disclosed
US-20110012100-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2011-01-20 US disclosed
EP-2254896-A1 METAL COMPLEXES Merck Patent GmbH (DE) 2010-12-01 EP disclosed
US-20100227978-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2010-09-09 US disclosed
US-7728137-B2 Metal complexes MERCK PATENT GMBH (DE) 2010-06-01 US disclosed
WO-2009118087-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2009-10-01 WO disclosed
EP-1603923-B9 METAL COMPLEXES MERCK PATENT GMBH (DE) 2007-10-31 EP disclosed
EP-1603923-A1 METAL COMPLEXES Covion Organic Semiconductors GmbH (DE) 2005-12-14 EP disclosed
WO-2004081017-A1 METAL COMPLEXES COVION ORGANIC SEMICONDUCTORS GMBH (DE) 2004-09-23 WO disclosed
US-6281303-B1 TRANSITION METAL COMPLEX EASTMAN CHEMICAL COMPANY 2001-08-28 US disclosed
US-5861140-A Tripodal paramagnetic contrast agents for MR imaging HOECHST CELANESE CORP. (US) 1999-01-19 US disclosed
US-5861138-A Ligands for MRI contrast agent HOECHST CELANESE CORP. (US) 1999-01-19 US disclosed
US-5858329-A MRI diagnostic procedures using tripodal pyridinyl metal complexes HOECHST CELANESE CORPORATION (US) 1999-01-12 US disclosed
US-5824288-A CONTRAST AGENTS FOR MAGNETIC RESONANCE IMAGING HOECHST CELANESE CORPORATION (US) 1998-10-20 US disclosed
US-5820851-A MAGNETIC RESONANCE IMAGING; RESOLUTION HOECHST CELANESE CORPORATION (US) 1998-10-13 US disclosed
WO-1998022148-A1 MRI CONTRAST AGENTS AND LIGANDS WASHINGTON UNIVERSITY (US) 1998-05-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100227978-A1 METAL COMPLEXES AP1M1, SOD1, AP2M1 HTR7 4647/4885HTR1A 3446/4885DRD2 3076/4885
US-20110012100-A1 METAL COMPLEXES AP1M1, AP3M1, SOD1 HTR7 4447/4885HTR1A 4297/4885DRD2 4278/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.