SCHEMBL9561804

SCHEMBL9561804

O=C(NCc1cccc(Cl)c1)c1ccnc(C(=O)[NH+]([O-])Cc2cccc(Cl)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
MAPK3 P27361 1/20 0.48
MAPK1 P28482 1/20 0.48
MMP13 P45452 1/20 0.46
ROCK2 O75116 3/20 0.46
RAB9A P51151 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ROCK1 Q13464 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA2B P29275 1/20 0.44
ADORA1 P30542 1/20 0.44
HPGD P15428 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214954 0.85 NPC1 (0.63) NPC1MAPK3MAPK1MMP13ROCK2
SCHEMBL9561684 0.79 KDM1A (0.53) MMP13ROCK2KMT2AGAASMN1; SMN2
SCHEMBL5216536 0.76 KMT2A (0.65) NPC1MAPK1ROCK2RAB9AHPGD
SCHEMBL1569143 0.75 NPC1 (0.73) NPC1MAPK3MAPK1ROCK2CYP2D6
SCHEMBL5332860 0.75 NPC1 (0.72) NPC1MAPK3MAPK1MMP13RAB9A
SCHEMBL5214984 0.74 CYP1A2 (0.50) NPC1MMP13ROCK2CYP1A2CYP2C9
SCHEMBL1767368 0.73 NPC1 (0.59) NPC1MAPK3MAPK1RAB9ACYP1A2
SCHEMBL5213178 0.71 CYP1A2 (0.64) MAPK1MMP13RAB9ACYP1A2CYP2C9
SCHEMBL8358422 0.71 MMP13 (0.68) NPC1MAPK1MMP13ROCK2RAB9A
SCHEMBL5213782 0.71 ROCK2 (0.58) MMP13ROCK2ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260323-A 2,4- and 2,5-substituted pyridine-N-oxides, processes for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-09 US disclosed