SCHEMBL9561684

SCHEMBL9561684

Cc1ccc(CNC(=O)c2ccnc(C(=O)[NH+]([O-])Cc3ccc(C)cc3)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.53
HDAC1 Q13547 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.50
POLB P06746 1/20 0.50
HTT P42858 3/20 0.47
LMNA P02545 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
KMT2A Q03164 1/20 0.45
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
ROCK2 O75116 1/20 0.43
MMP2 P08253 1/20 0.43
CYP3A4 P08684 1/20 0.43
STAT3 P40763 1/20 0.43
MMP13 P45452 1/20 0.43
MAPK14 Q16539 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212608 0.84 SMN1; SMN2 (0.64) KDM1AHDAC1SMN1; SMN2POLBHTT
SCHEMBL9561804 0.79 NPC1 (0.53) SMN1; SMN2KMT2AGAAROCK2MMP13
SCHEMBL5213342 0.74 RAB9A (0.60) SMN1; SMN2HTTLMNAKMT2AMAPT
SCHEMBL1568232 0.72 SMN1; SMN2 (0.74) SMN1; SMN2POLBHTTLMNAL3MBTL1
SCHEMBL5215174 0.71 EPHX2 (0.52) KDM1AHDAC1SMN1; SMN2POLBHTT
SCHEMBL14256291 0.71 L3MBTL1 (0.67) KDM1AHDAC1SMN1; SMN2POLBHTT
SCHEMBL5213178 0.71 CYP1A2 (0.64) SMN1; SMN2POLBHTTLMNAKMT2A
SCHEMBL5212711 0.71 RAB9A (0.67) KDM1AHDAC1SMN1; SMN2POLBL3MBTL1
SCHEMBL8358422 0.71 MMP13 (0.68) SMN1; SMN2HTTLMNAL3MBTL1ALDH1A1
SCHEMBL5209755 0.71 SMN1; SMN2 (0.64) SMN1; SMN2HTTLMNAL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260323-A 2,4- and 2,5-substituted pyridine-N-oxides, processes for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-09 US disclosed